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9YLH

Human p38 ALPHA MAPK:MW01-8-105SRM N,N-Dimethyl-6-phenyl-5-(4-pyridinyl)-3-pyridazinamine inhibitor complex

This is a non-PDB format compatible entry.
Summary for 9YLH
Entry DOI10.2210/pdb9ylh/pdb
DescriptorMitogen-activated protein kinase 14, ZINC ION, 4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDINE, ... (5 entities in total)
Functional Keywordsserine/threonine-protein kinase, protein kinase domain, transferase, atp binding, phosphorylation, cytosol, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight42080.29
Authors
Brunzelle, J.S.,Shuvalova, L.,Roy, S.M.,Watterson, D.M. (deposition date: 2025-10-08, release date: 2025-11-19)
Primary citationBrunzelle, J.S.,Shuvalova, L.,Roy, S.M.,Watterson, D.M.
Human p38 ALPHA MAPK:MW01-8-105SRM N,N-Dimethyl-6-phenyl-5-(4-pyridinyl)-3-pyridazinamine inhibitor complex
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.02 Å)
Structure validation

247947

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