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9WN9

Wild-type Menin complexed with DSP-5336

Summary for 9WN9
Entry DOI10.2210/pdb9wn9/pdb
DescriptorMenin, 5-fluoro-2-[(4-{7-[(1S,3S,4R)-5-methylidene-2-azabicyclo[2.2.2]octane-3-carbonyl]-2,7-diazaspiro[3.5]nonan-2-yl}pyrimidin-5-yl)oxy]-N,N-di(propan-2-yl)benzamide, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordshuman menin, transcription, m322i mutant inhibitor complex, ds1594
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight111051.71
Authors
Bijpuria, S.,Mckeever, B.M.,Mcgeehan, G.M. (deposition date: 2025-09-04, release date: 2026-04-29, Last modification date: 2026-05-13)
Primary citationBijpuria, S.,Mckeever, B.M.,Mcgeehan, G.M.
Wild-type Menin complexed with DSP-5336
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

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PDB entries from 2026-07-22

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