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9WKW

Wild-type Menin complexed with DS-1594

Summary for 9WKW
Entry DOI10.2210/pdb9wkw/pdb
Related7UJ4
DescriptorMenin, (1R,2S,4R)-4-[[4-(5,6-dimethoxypyridazin-3-yl)phenyl]methylamino]-2-[methyl-[6-[2,2,2-tris(fluoranyl)ethyl]thieno[2,3-d]pyrimidin-4-yl]amino]cyclopentan-1-ol, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordshuman menin, transcription, m322i mutant inhibitor complex, sndx-5613
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight111596.66
Authors
Bijpuria, S.,Mckeever, B.M.,Mcgeehan, G.M. (deposition date: 2025-09-01, release date: 2026-04-29)
Primary citationBijpuria, S.,Mckeever, B.M.,Mcgeehan, G.M.
Wild-type Menin complexed with DS-1594
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.63 Å)
Structure validation

257629

PDB entries from 2026-08-05

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