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9SIZ

CK1d in complex with IG138

This is a non-PDB format compatible entry.
Summary for 9SIZ
Entry DOI10.2210/pdb9siz/pdb
DescriptorCasein kinase I isoform delta, 5-(4-fluorophenyl)-~{N}2-piperidin-4-yl-6-pyridin-4-yl-pyrazine-2,3-diamine, MALONATE ION, ... (5 entities in total)
Functional Keywordskinase inhibitors, ck1delta, pyrazines, als, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight69928.77
Authors
Trevisan, L.,Morasso, S.,Dalle Vedove, A.,Spalluto, G.,Storici, P.,Federico, S. (deposition date: 2025-08-29, release date: 2026-09-09)
Primary citationTrevisan, L.,Morasso, S.,Dalle Vedove, A.,Spalluto, G.,Storici, P.,Federico, S.
Crystal structures of CK1d with pyrazine inhibitors
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

260626

PDB entries from 2026-10-07

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