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9SIX

CK1d in complex with IG130

This is a non-PDB format compatible entry.
Summary for 9SIX
Entry DOI10.2210/pdb9six/pdb
DescriptorCasein kinase I isoform delta, 6-(4-fluorophenyl)-3-(4-methylpiperazin-1-yl)-5-pyridin-4-yl-pyrazin-2-amine, MALONATE ION, ... (5 entities in total)
Functional Keywordskinase inhibitors, ck1delta, pyrazines, als, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight70092.88
Authors
Trevisan, L.,Morasso, S.,Dalle Vedove, A.,Spalluto, G.,Storici, P.,Federico, S. (deposition date: 2025-08-29, release date: 2026-09-09)
Primary citationTrevisan, L.,Morasso, S.,Dalle Vedove, A.,Spalluto, G.,Storici, P.,Federico, S.
Crystal structures of CK1d with pyrazine inhibitors
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.23 Å)
Structure validation

260320

PDB entries from 2026-09-30

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