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9RLW

Leishmania major N-myristoyltransferase in complex with azetidinopyrimidine inhibitor IMP-825

This is a non-PDB format compatible entry.
Summary for 9RLW
Entry DOI10.2210/pdb9rlw/pdb
Related6B1L
DescriptorGlycylpeptide N-tetradecanoyltransferase, MAGNESIUM ION, ~{N}-[[2,4-bis(fluoranyl)phenyl]methyl]-1-[5-chloranyl-2-[2-(dimethylamino)ethylamino]pyrimidin-4-yl]azetidine-3-carboxamide, ... (5 entities in total)
Functional Keywordsmyristoylation, azetidinopyrimidine, leishmania, inhibitor, transferase
Biological sourceLeishmania major
Total number of polymer chains1
Total formula weight49622.84
Authors
Brannigan, J.A. (deposition date: 2025-06-17, release date: 2026-05-27)
Primary citationBell, A.S.
Leishmania major N-myristoyltransferase in complex with azetidinopyrimidine inhibitor IMP-825
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.49 Å)
Structure validation

255239

PDB entries from 2026-06-17

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