9RLU

Leishmania major N-myristoyltransferase in complex with azetidinopyrimidine inhibitor IMP-819

This is a non-PDB format compatible entry.

Summary for 9RLU

• Entry DOI: 10.2210/pdb9rlu/pdb
• Related: 6B1L
• Descriptor: Glycylpeptide N-tetradecanoyltransferase, TETRADECANOYL-COA, 1-[5-chloranyl-2-[2-(dimethylamino)ethylamino]pyrimidin-4-yl]-~{N}-[(5-methylpyrazin-2-yl)methyl]azetidine-3-carboxamide, ... (5 entities in total)
• Functional Keywords: myristoylation, azetidinopyrimidine, leishmania, inhibitor, transferase
• Biological source: Leishmania major
• Total number of polymer chains: 1
• Total formula weight: 49602.86

Authors

Brannigan, J.A. (deposition date: 2025-06-17, release date: 2026-05-27)

• Primary citation: Bell, A.S.; Leishmania major N-myristoyltransferase in complex with azetidinopyrimidine inhibitor IMP-819; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.3 Å)