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9QST

Protein Kinase CK2 and bivalent inhibitors

This is a non-PDB format compatible entry.
Summary for 9QST
Entry DOI10.2210/pdb9qst/pdb
DescriptorCasein kinase II subunit alpha, SULFATE ION, 5-[4-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanoylamino]butylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid, ... (4 entities in total)
Functional Keywordsprotein kinase inhibitor bivalent ad pocket, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight87628.02
Authors
Krimm, I.,Gelin, M.,Guichou, J.F.,Grenier, D. (deposition date: 2025-04-07, release date: 2026-04-15)
Primary citationKrimm, I.,Gelin, M.,Guichou, J.F.,Grenier, D.
Protein Kinase CK2 and bivalent inhibitors
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.7 Å)
Structure validation

254917

PDB entries from 2026-06-10

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