9QNV

CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound 2

This is a non-PDB format compatible entry.

Summary for 9QNV

• Entry DOI: 10.2210/pdb9qnv/pdb
• Descriptor: Bromodomain-containing protein 4, 1,2-ETHANEDIOL, 3-methyl-5-phenyl-[1,3]thiazolo[2,3-c][1,2,4]triazole, ... (5 entities in total)
• Functional Keywords: bromodomain-containing protein 4 isoform long, brd4, bromodomain-containing protein 4, cap, hunk1, mcap, mitotic chromosome associated protein, cell cycle, structural genomics, structural genomics consortium, sgc
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 15602.02

Authors

Krojer, T.,Martinez-Cartro, M.,Picaud, S.,Filippakopoulos, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Barril, X.,von Delft, F.,Structural Genomics Consortium (SGC) (deposition date: 2025-03-25, release date: 2025-05-14)

• Primary citation: Krojer, T.,Martinez-Cartro, M.,Picaud, S.,Filippakopoulos, P.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Barril, X.,von Delft, F.; CRYSTAL STRUCTURE OF THE FIRST BROMODOMAIN OF HUMAN BRD4 IN COMPLEX with compound 2; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.226 Å)