9NTZ
Crystal structure of calcium-dependent protein kinase 1 (CDPK1) from Cryptosporidium parvum in complex with inhibitor BKI-1932.
This is a non-PDB format compatible entry.
Summary for 9NTZ
| Entry DOI | 10.2210/pdb9ntz/pdb |
| Descriptor | Calmodulin-domain protein kinase 1, (6R,8M)-8-(2-ethoxyquinolin-6-yl)-5,5-dimethyl-2-oxo-1,2,4,5-tetrahydropyrazolo[5,1-d][1,3,5]oxadiazepine-9-carboxamide, L(+)-TARTARIC ACID, ... (5 entities in total) |
| Functional Keywords | ssgcid, structural genomics, seattle structural genomics center for infectious disease, transferase, cryptosporidium parvum, cdpk1 |
| Biological source | Cryptosporidium parvum Iowa II |
| Total number of polymer chains | 1 |
| Total formula weight | 57416.20 |
| Authors | Seattle Structural Genomics Center for Infectious Disease,Seattle Structural Genomics Center for Infectious Disease (SSGCID) (deposition date: 2025-03-19, release date: 2026-04-01) |
| Primary citation | Liu, L.,Lovell, S.,Battaile, K.P. Crystal structure of calcium-dependent protein kinase 1 (CDPK1) from Cryptosporidium parvum in complex with inhibitor BKI-1932. To be published, |
| Experimental method | X-RAY DIFFRACTION (1.84 Å) |
Structure validation
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