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9MRQ

Mycobacterium tuberculosis RNA polymerase elongation complex bound to inhibitor N-aroyl-N-aryl-phenylalanine amide (AAP)-SO2

This is a non-PDB format compatible entry.
Summary for 9MRQ
Entry DOI10.2210/pdb9mrq/pdb
EMDB information48561
DescriptorDNA-directed RNA polymerase subunit alpha, MAGNESIUM ION, DNA-directed RNA polymerase subunit beta, ... (11 entities in total)
Functional Keywordsrna polymerase, transcription, transferase-inhibitor complex, elongation, transcription inhibitor, transferase/inhibitor
Biological sourceMycobacterium tuberculosis H37Rv
More
Total number of polymer chains8
Total formula weight404729.50
Authors
Bosch, B.,Lilic, M.,Campbell, E.A. (deposition date: 2025-01-08, release date: 2025-10-08)
Primary citationBarbara, B.,Lilic, M.,Campbell, E.A.
Co-inhibition of Transcription Reduces Rifampicin Resistance and Enhances Killing of Mycobacterium tuberculosis.
To Be Published,
Experimental method
ELECTRON MICROSCOPY (2.97 Å)
Structure validation

247536

PDB entries from 2026-01-14

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