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9KXT

Structure of human B0AT1-ACE2 complex with compound1

This is a non-PDB format compatible entry.
Summary for 9KXT
Entry DOI10.2210/pdb9kxt/pdb
EMDB information62627
DescriptorSodium-dependent neutral amino acid transporter B(0)AT1, Angiotensin-converting enzyme 2, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (6 entities in total)
Functional Keywordsinhibitor, amino acid transporter, slc6, transport protein
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight166905.01
Authors
Imazu, T.,Miyaguchi, I.,Hiraizumi, M. (deposition date: 2024-12-07, release date: 2025-12-10)
Primary citationImazu, T.,Akashi, T.,Hiraizumi, M.,Inui, Y.,Sasaki, W.,Takahashi, T.,Todoroki, H.,Kumanomidou, T.,Hisano, H.,Asada, H.,Kusakizako, T.,Nishizawa, T.,Iwata, S.,Nureki, O.,Miyaguchi, I.
Structure-guided development of a potent human B0AT1 inhibitor effective in a mouse model of phenylketonuria
To Be Published,
Experimental method
ELECTRON MICROSCOPY (2.7 Å)
Structure validation

247536

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