9KVW

Crystal Structures of Keap1-compound complexes

This is a non-PDB format compatible entry.

Summary for 9KVW

• Entry DOI: 10.2210/pdb9kvw/pdb
• Descriptor: Kelch-like ECH-associated protein 1, ~{N}-[4-[(2-azanyl-2-oxidanylidene-ethyl)-[4-[(2-azanyl-2-oxidanylidene-ethyl)-(4-methoxyphenyl)sulfonyl-amino]naphthalen-1-yl]sulfamoyl]phenyl]-3-(2-oxa-8-azaspiro[4.5]decan-8-yl)propanamide (3 entities in total)
• Functional Keywords: complex, inhibitor, protein binding
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 32376.22

Authors

Zhuang, C.L.,Yu, R.L. (deposition date: 2024-12-05, release date: 2025-12-10)

• Primary citation: Zhuang, C.L.,Yu, R.Z.; Crystal structure of Keap1-CD10; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.44 Å)