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9KSA

Serine Beta-Lactamase OXA-48 in Complex with MBL/SBL Inhibitor CB1

This is a non-PDB format compatible entry.
Summary for 9KSA
Entry DOI10.2210/pdb9ksa/pdb
DescriptorBeta-lactamase, 2-oxidanyl-7-(pyrazol-1-ylmethyl)-3~{H}-1,4,2-benzodioxaborinine-8-carboxylic acid (3 entities in total)
Functional Keywordsbeta-lactamase, serine-beta-lactamase oxa-48, oxa-48, hydrolase
Biological sourceKlebsiella pneumoniae
Total number of polymer chains4
Total formula weight113487.23
Authors
Li, G.-B.,Wei, S.-Q. (deposition date: 2024-11-29, release date: 2025-09-03)
Primary citationLi, G.-B.,Wei, S.-Q.
OXA-48 carbapenemase in complex with 7-((1H-pyrazol-1-yl)methyl)-2-hydroxy-2,3-dihydrobenzo[e][1,4,2]dioxaborinine-8-carboxylic acid
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.178 Å)
Structure validation

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