Summary for 9KQY
| Entry DOI | 10.2210/pdb9kqy/pdb |
| Descriptor | Dual specificity tyrosine-phosphorylation-regulated kinase 2, [6-[[4-[2-(diethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-propan-2-ylpiperazin-1-yl)methanone (2 entities in total) |
| Functional Keywords | dyrk2, tsl2109, cell cycle |
| Biological source | Homo sapiens (human) |
| Total number of polymer chains | 2 |
| Total formula weight | 94313.11 |
| Authors | Tong, C. (deposition date: 2024-11-27, release date: 2025-12-03, Last modification date: 2025-12-17) |
| Primary citation | Tong, C. The co-crystal structure of DYRK2 with TSL2109 To Be Published, |
| Experimental method | X-RAY DIFFRACTION (3.2 Å) |
Structure validation
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