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9KQY

The co-crystal structure of DYRK2 with TSL2109

This is a non-PDB format compatible entry.
Summary for 9KQY
Entry DOI10.2210/pdb9kqy/pdb
DescriptorDual specificity tyrosine-phosphorylation-regulated kinase 2, [6-[[4-[2-(diethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-propan-2-ylpiperazin-1-yl)methanone (2 entities in total)
Functional Keywordsdyrk2, tsl2109, cell cycle
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight94313.11
Authors
Tong, C. (deposition date: 2024-11-27, release date: 2025-12-03, Last modification date: 2025-12-17)
Primary citationTong, C.
The co-crystal structure of DYRK2 with TSL2109
To Be Published,
Experimental method
X-RAY DIFFRACTION (3.2 Å)
Structure validation

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