Summary for 9I9U
| Entry DOI | 10.2210/pdb9i9u/pdb |
| Descriptor | Histone-arginine methyltransferase CARM1, (phenylmethyl) (2S)-5-[(Z)-[[3-[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]propylamino]-(methylamino)methylidene]amino]-2-(phenylmethoxycarbonylamino)pentanoate, CHLORIDE ION, ... (4 entities in total) |
| Functional Keywords | protein arginine n-methyltransferase, prmt, carm1, transition state mimics, transcription, transferase |
| Biological source | Mus musculus (house mouse) |
| Total number of polymer chains | 4 |
| Total formula weight | 170737.05 |
| Authors | Cura, V.,Dursun, E.,Troffer, N.,Cavarelli, J. (deposition date: 2025-02-07, release date: 2026-02-18) |
| Primary citation | Cura, V.,Dursun, E.,Troffer, N.,Cavarelli, J. CARM1 in complex with arg-aDMA analog To Be Published, |
| Experimental method | X-RAY DIFFRACTION (2.2 Å) |
Structure validation
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