9GZD
Androgen Receptor ligand-binding domain in complex with 11-ketodihydrotestosterone
This is a non-PDB format compatible entry.
Summary for 9GZD
| Entry DOI | 10.2210/pdb9gzd/pdb |
| Descriptor | Androgen receptor, 11-ketodihydrotestosterone, SPERMIDINE, ... (7 entities in total) |
| Functional Keywords | nulcear receptor, hormone binding, prostate cancer, dna binding protein |
| Biological source | Homo sapiens (human) |
| Total number of polymer chains | 1 |
| Total formula weight | 29845.08 |
| Authors | Alegre-Marti, A.,Zwart, W.,Fuentes-Prior, P.,Estebanez-Perpina, E. (deposition date: 2024-10-03, release date: 2026-04-15) |
| Primary citation | Minnee, E.,Lacoste, A.,Alegre-Marti, A.,Gregoricchio, S.,Fuentes-Prior, P.,van der Zande, K.,van Herwaarden, T.,Estebanez-Perpina, E.,Bergman, A.M.,Zwart, W. Multi-omics and structural analyses on Androgen Receptor reveals highly similar biological actions of testosterone variants from testicular versus adrenal origins in prostate cancer cells To Be Published, |
| Experimental method | X-RAY DIFFRACTION (1.91 Å) |
Structure validation
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