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9FLO

Crystal structure of human Haspin (GSG2) kinase bound to MU2181

This is a non-PDB format compatible entry.
Summary for 9FLO
Entry DOI10.2210/pdb9flo/pdb
DescriptorSerine/threonine-protein kinase haspin, NICKEL (II) ION, ~{N}-(1,4-dimethylpyrazol-3-yl)-3-(1,2-thiazol-5-yl)thieno[3,2-b]pyridin-5-amine, ... (4 entities in total)
Functional Keywordshaspin, kinase, inhibitor, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight41097.60
Authors
Kraemer, A.,Paruch, K.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2024-06-05, release date: 2024-09-11)
Primary citationKraemer, A.,Paruch, K.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of human Haspin (GSG2) kinase bound to MU2181
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.9 Å)
Structure validation

225946

PDB entries from 2024-10-09

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