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9EQ0

Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with allosteric ligand FGJG12

This is a non-PDB format compatible entry.
Summary for 9EQ0
Entry DOI10.2210/pdb9eq0/pdb
DescriptorCasein kinase II subunit alpha, SULFATE ION, ~{N}-[4-[(3-chloranyl-4-phenyl-phenyl)methylamino]butyl]isoquinoline-5-sulfonamide, ... (4 entities in total)
Functional Keywordsck2, kinase, chemical, allosteric inhibitor, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight82192.38
Authors
Kraemer, A.,Greco, F.,Gerninghaus, J.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2024-03-20, release date: 2024-05-01)
Primary citationKraemer, A.,Greco, F.,Gerninghaus, J.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with allosteric ligand FGJG12
To Be Published,
Experimental method
X-RAY DIFFRACTION (3.15 Å)
Structure validation

220113

PDB entries from 2024-05-22

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