9D04
CO-CRYSTAL STRUCTURE OF CIRCULARLY PERMUTED HUMAN TASPASE-1 BOUND TO LIGAND SMDC994967 1-(ETHENESULFONYL)-4-{[4- (TRIFLUOROMETHOXY)PHENYL]METHYL}PIPERAZINE
Summary for 9D04
| Entry DOI | 10.2210/pdb9d04/pdb |
| Related | 6VKW |
| Descriptor | Threonine aspartase subunit beta,Threonine aspartase subunit alpha, SODIUM ION, CHLORIDE ION, ... (5 entities in total) |
| Functional Keywords | mll, taspase-1, circular permutation, hydrolase |
| Biological source | Homo sapiens (human) More |
| Total number of polymer chains | 2 |
| Total formula weight | 71540.98 |
| Authors | |
| Primary citation | Delker, S.L.,Edwards, T.E.,Abendroth, J. CO-CRYSTAL STRUCTURE OF CIRCULARLY PERMUTED HUMAN TASPASE-1 BOUND TO LIGAND SMDC994967 1-(ETHENESULFONYL)-4-{[4- (TRIFLUOROMETHOXY)PHENYL]METHYL}PIPERAZINE TO BE PUBLISHED, |
| Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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