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9D04

CO-CRYSTAL STRUCTURE OF CIRCULARLY PERMUTED HUMAN TASPASE-1 BOUND TO LIGAND SMDC994967 1-(ETHENESULFONYL)-4-{[4- (TRIFLUOROMETHOXY)PHENYL]METHYL}PIPERAZINE

Summary for 9D04
Entry DOI10.2210/pdb9d04/pdb
Related6VKW
DescriptorThreonine aspartase subunit beta,Threonine aspartase subunit alpha, SODIUM ION, CHLORIDE ION, ... (5 entities in total)
Functional Keywordsmll, taspase-1, circular permutation, hydrolase
Biological sourceHomo sapiens (human)
More
Total number of polymer chains2
Total formula weight71540.98
Authors
Delker, S.L.,Edwards, T.E.,Abendroth, J. (deposition date: 2024-08-06, release date: 2025-08-13)
Primary citationDelker, S.L.,Edwards, T.E.,Abendroth, J.
CO-CRYSTAL STRUCTURE OF CIRCULARLY PERMUTED HUMAN TASPASE-1 BOUND TO LIGAND SMDC994967 1-(ETHENESULFONYL)-4-{[4- (TRIFLUOROMETHOXY)PHENYL]METHYL}PIPERAZINE
TO BE PUBLISHED,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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