9CKP

Human G protein-coupled receptor kinase 5-D311N in complex with sangivamycin

Summary for 9CKP

• Entry DOI: 10.2210/pdb9ckp/pdb
• Descriptor: G protein-coupled receptor kinase 5, ACETYL GROUP, SANGIVAMYCIN, ... (5 entities in total)
• Functional Keywords: gpcr, grk, g protein-coupled receptor, g protein-coupled receptor kinase, gpcr signaling, signaling protein
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 69324.16

Authors

Chen, Y.,Tesmer, J.J.G. (deposition date: 2024-07-09, release date: 2025-07-16)

• Primary citation: Chen, Y.,Tesmer, J.J.G.; Structures of G protein-coupled receptor kinase 5 in multiple conformations reveals mechanism of activation and inhibition; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.6 Å)