8TZI

Human equilibrative nucleoside transporter-1, JH-ENT-01 bound

8TZI の概要

• エントリーDOI: 10.2210/pdb8tzi/pdb
• 分子名称: Equilibrative nucleoside transporter 1, (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, 3-[4-[3-[3,4-dimethoxy-5-[[4-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methoxy]phenyl]carbonyloxypropyl]-1,4-diazepan-1-yl]propyl 3,4,5-trimethoxybenzoate, ... (4 entities in total)
• 機能のキーワード: adenosine transport, adenosine reuptake inhibitor, nucleoside, hent1, equilibrative nucleoside transporter, slc29, transport protein-inhibitor complex, transport protein/inhibitor
• 由来する生物種: Homo sapiens (human)
• タンパク質・核酸の鎖数: 1
• 化学式量合計: 51729.74

構造登録者

Wright, N.J.,Lee, S.Y. (登録日: 2023-08-26, 公開日: 2024-08-28)

• 主引用文献: Wright, N.J.,Lee, S.Y.; Rational ENT1 inhibition as a pathway for neuropathic pain relief; To Be Published,

実験手法

X-RAY DIFFRACTION (2.7 Å)