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8R7W

Kras G12D in complex with compound 3

Summary for 8R7W
Entry DOI10.2210/pdb8r7w/pdb
DescriptorGTPase KRas, PHOSPHOMETHYLPHOSPHONIC ACID GUANYLATE ESTER, 8-(furan-3-yl)-2,3,4,9-tetrahydropyrido[3,4-b]indol-1-one, ... (5 entities in total)
Functional Keywordskras, inhibitor, small molecule compound, oncoprotein
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight40369.26
Authors
Zak, K.M.,Kessler, D. (deposition date: 2023-11-27, release date: 2024-10-02)
Primary citationZak, K.M.,Kessler, D.
Kras G12D in complex with compound 3
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.161 Å)
Structure validation

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PDB entries from 2024-10-02

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