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8QWZ

Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 4-(6-(6-isopropoxy-1H-indol-1-yl)pyrazin-2-yl)benzoic acid

Summary for 8QWZ
Entry DOI10.2210/pdb8qwz/pdb
DescriptorCasein kinase II subunit alpha, SULFATE ION, 4-[6-(6-propan-2-yloxyindol-1-yl)pyrazin-2-yl]benzoic acid, ... (4 entities in total)
Functional Keywordsck2, inhibitor, kinase, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight82459.46
Authors
Kraemer, A.,Galal, K.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2023-10-20, release date: 2024-01-17)
Primary citationKraemer, A.,Galal, K.,Willson, T.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of human Casein Kinase II subunit alpha (CK2a1) in complex with 4-(6-(6-isopropoxy-1H-indol-1-yl)pyrazin-2-yl)benzoic acid
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.6 Å)
Structure validation

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PDB entries from 2024-04-24

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