8QQG
Structure of BRAF in Complex With Exarafenib (KIN-2787).
Summary for 8QQG
Entry DOI | 10.2210/pdb8qqg/pdb |
Descriptor | Serine/threonine-protein kinase B-raf, (3~{S})-~{N}-[4-methyl-3-[2-morpholin-4-yl-6-[[(2~{R})-1-oxidanylpropan-2-yl]amino]pyridin-4-yl]phenyl]-3-[2,2,2-tris(fluoranyl)ethyl]pyrrolidine-1-carboxamide, CHLORIDE ION, ... (4 entities in total) |
Functional Keywords | transferase, braf |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 3 |
Total formula weight | 95866.88 |
Authors | Schmitt, A.,Costanzi, E.,Kania, R.,Chen, Y.K. (deposition date: 2023-10-04, release date: 2024-01-24) |
Primary citation | Schmitt, A.,Costanzi, E.,Kania, R.,Chen, Y.K. Structure of BRAF in Complex With Exarafenib (KIN-2787). To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.979 Å) |
Structure validation
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