8PIQ
Crystal Structure of BRD4-BD1 with BI894999
Summary for 8PIQ
Entry DOI | 10.2210/pdb8piq/pdb |
Descriptor | Bromodomain-containing protein 4, ~{N},3-dimethyl-6-[6-(4-methylpiperazin-1-yl)-1-(phenylmethyl)benzimidazol-2-yl]-[1,2,4]triazolo[4,3-a]pyrazin-8-amine, 1,2-ETHANEDIOL, ... (5 entities in total) |
Functional Keywords | boehringeringelheim, brd4, inhibitor, transcription |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 15769.22 |
Authors | Kessler, D. (deposition date: 2023-06-22, release date: 2023-07-26, Last modification date: 2024-06-19) |
Primary citation | Kessler, D. Crystal Structure of BRD4-BD1 with BI894999 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.117 Å) |
Structure validation
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