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8PAI

Crystal structure of human Histidine Triad Nucleotide-Binding Protein 1 in complex with 5'-O-[N-(3-Indolepropionic acid)sulfamoyl] N2-methyl-2-aminoethenoadenosine

Summary for 8PAI
Entry DOI10.2210/pdb8pai/pdb
DescriptorHistidine triad nucleotide-binding protein 1, 5'-O-[N-(3-Indolepropionic acid)sulfamoyl] N2-methyl-2-aminoethenoadenosine (3 entities in total)
Functional Keywordshint, hit, histidine triad, phosphoramidase, complex, inhibitor, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight28218.44
Authors
Dolot, R.M.,Dillenburg, M.,Wagner, C.R. (deposition date: 2023-06-07, release date: 2023-06-14, Last modification date: 2024-06-19)
Primary citationDillenburg, M.,Dolot, R.,Wagner, C.R.
Novel inhibitors for hHINT1 protein
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

222415

PDB entries from 2024-07-10

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