8P9B
Crystal Structure of Mnk2-D228G in complex with Tinodasertib
Summary for 8P9B
Entry DOI | 10.2210/pdb8p9b/pdb |
Descriptor | MAP kinase-interacting serine/threonine-protein kinase 2, ZINC ION, 4-[6-(4-morpholin-4-ylcarbonylphenyl)imidazo[1,2-a]pyridin-3-yl]benzenecarbonitrile (3 entities in total) |
Functional Keywords | mnk2, transferase-transferase inhibitor complex, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 36078.32 |
Authors | Turnbull, A.P.,Sabin, V.,Bell, C.,Watson, M. (deposition date: 2023-06-05, release date: 2024-06-12) |
Primary citation | Sabin, V.,Turnbull, A.P.,Bell, C.,Watson, M. Crystal Structure of Mnk2-D228G in complex with Tinodasertib To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.59 Å) |
Structure validation
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