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8P9B

Crystal Structure of Mnk2-D228G in complex with Tinodasertib

Summary for 8P9B
Entry DOI10.2210/pdb8p9b/pdb
DescriptorMAP kinase-interacting serine/threonine-protein kinase 2, ZINC ION, 4-[6-(4-morpholin-4-ylcarbonylphenyl)imidazo[1,2-a]pyridin-3-yl]benzenecarbonitrile (3 entities in total)
Functional Keywordsmnk2, transferase-transferase inhibitor complex, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight36078.32
Authors
Turnbull, A.P.,Sabin, V.,Bell, C.,Watson, M. (deposition date: 2023-06-05, release date: 2024-06-12)
Primary citationSabin, V.,Turnbull, A.P.,Bell, C.,Watson, M.
Crystal Structure of Mnk2-D228G in complex with Tinodasertib
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.59 Å)
Structure validation

224004

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