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8P1F

X-ray structure of acetylcholine-binding protein (AChBP) in complex with FL001909.

Summary for 8P1F
Entry DOI10.2210/pdb8p1f/pdb
DescriptorAcetylcholine-binding protein, 2-acetamido-2-deoxy-beta-D-glucopyranose, 4-azanyl-1-phenyl-piperidine-4-carboxylic acid, ... (4 entities in total)
Functional Keywordsfragment based drug design, acetylcholine-binding protein, choline-binding proteins, choline-binding protein
Biological sourceLymnaea stagnalis (great pond snail)
Total number of polymer chains20
Total formula weight544742.91
Authors
Primary citationFitzgerald, E.A.,Cederfelt, D.,Boronat, P.,Aarmo Lund, B.,de Esch, I.J.P.,Danielson, U.H.
Elucidating the regulation of ligand gated ion channels via biophysical studies of ligand-induced conformational dynamics of acetylcholine binding proteins
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

219869

PDB entries from 2024-05-15

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