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8OKT

Carbonic Anhydrase IX like mutant in Complex with Steriod_Sulphamoyl inhibitor VK42

Summary for 8OKT
Entry DOI10.2210/pdb8okt/pdb
DescriptorCarbonic anhydrase 2, ZINC ION, [(8~{R},9~{S},13~{S},14~{S})-13-methyl-17-oxidanylidene-7,8,9,11,12,14,15,16-octahydro-6~{H}-cyclopenta[a]phenanthren-3-yl] sulfamate, ... (4 entities in total)
Functional Keywordscarbonic anhydrase, inhibitor, oncoprotein
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight29643.76
Authors
Brynda, J.,Rezacova, P.M.,Kudova, E. (deposition date: 2023-03-29, release date: 2024-04-10)
Primary citationBrynda, J.,Rezacova, P.M.,Kudova, E.
Carbonic Anhydrase II in Complex with Steriod_Sulphamoyl
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

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PDB entries from 2024-04-24

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