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8OKP

Carbonic Anhydrase IX like mutant in Complex with Steriod_Sulphamoyl inhibitor AKI_33

Summary for 8OKP
Entry DOI10.2210/pdb8okp/pdb
DescriptorCarbonic anhydrase 2, ZINC ION, [(3~{R},5~{R},8~{R},9~{S},10~{S},13~{S},14~{S},15~{R})-10,13,15-trimethyl-17-oxidanylidene-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-3-yl] sulfamate, ... (4 entities in total)
Functional Keywordscarbonic anhydrase, inhibitor, oncoprotein
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight29649.84
Authors
Brynda, J.,Rezacova, P.M.,Kudova, E. (deposition date: 2023-03-28, release date: 2024-04-10)
Primary citationBrynda, J.,Rezacova, P.M.,Kudova, E.
Carbonic Anhydrase II in Complex with Steriod_Sulphamoyl
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.25 Å)
Structure validation

218853

PDB entries from 2024-04-24

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