8OF2
Trypanosoma brucei pteridine reductase 1 (TbPTR1) in complex with 2,4,6 triamminopyrimidine (TAP)
Summary for 8OF2
Entry DOI | 10.2210/pdb8of2/pdb |
Descriptor | Pteridine reductase, PYRIMIDINE-2,4,6-TRIAMINE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... (6 entities in total) |
Functional Keywords | trypanosoma brucei, pteridine reductase, ptr1, tbptr1, triamminopyrimidine, oxidoreductase |
Biological source | Trypanosoma brucei brucei |
Total number of polymer chains | 4 |
Total formula weight | 126341.53 |
Authors | |
Primary citation | Linciano, P.,Pozzi, C.,Tassone, G.,Landi, G.,Mangani, S.,Santucci, M.,Luciani, R.,Ferrari, S.,Santarem, N.,Tagliazucchi, L.,Cordeiro-da-Silva, A.,Tonelli, M.,Tondi, D.,Bertarini, L.,Gul, S.,Witt, G.,Moraes, C.B.,Costantino, L.,Costi, M.P. The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents. Eur.J.Med.Chem., 264:115946-115946, 2023 Cited by PubMed: 38043491DOI: 10.1016/j.ejmech.2023.115946 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.48 Å) |
Structure validation
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