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8OF2

Trypanosoma brucei pteridine reductase 1 (TbPTR1) in complex with 2,4,6 triamminopyrimidine (TAP)

Summary for 8OF2
Entry DOI10.2210/pdb8of2/pdb
DescriptorPteridine reductase, PYRIMIDINE-2,4,6-TRIAMINE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... (6 entities in total)
Functional Keywordstrypanosoma brucei, pteridine reductase, ptr1, tbptr1, triamminopyrimidine, oxidoreductase
Biological sourceTrypanosoma brucei brucei
Total number of polymer chains4
Total formula weight126341.53
Authors
Tassone, G.,Landi, G.,Mangani, S.,Pozzi, C. (deposition date: 2023-03-13, release date: 2023-12-13)
Primary citationLinciano, P.,Pozzi, C.,Tassone, G.,Landi, G.,Mangani, S.,Santucci, M.,Luciani, R.,Ferrari, S.,Santarem, N.,Tagliazucchi, L.,Cordeiro-da-Silva, A.,Tonelli, M.,Tondi, D.,Bertarini, L.,Gul, S.,Witt, G.,Moraes, C.B.,Costantino, L.,Costi, M.P.
The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents.
Eur.J.Med.Chem., 264:115946-115946, 2023
Cited by
PubMed: 38043491
DOI: 10.1016/j.ejmech.2023.115946
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.48 Å)
Structure validation

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