8JVE
Identification and characterization of inhibitors covalently modifying catalytic cysteine of UBE2T and blocking ubiquitin transfer
Summary for 8JVE
Entry DOI | 10.2210/pdb8jve/pdb |
Descriptor | Ubiquitin-conjugating enzyme E2 T, 1-(3-methoxyphenyl)-1,2,3,4-tetrazole, 1,2-ETHANEDIOL, ... (4 entities in total) |
Functional Keywords | ube2t, drug discovery, covalent inhibitor, fanconi anemia, ligase-inhibitor complex, ligase/inhibitor |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 18068.84 |
Authors | |
Primary citation | Anantharajan, J.,Tan, Q.W.,Fulwood, J.,Sifang, W.,Huang, Q.,Ng, H.Q.,Koh, X.,Xu, W.,Cherian, J.,Baburajendran, N.,Kang, C.,Ke, Z. Identification and characterization of inhibitors covalently modifying catalytic cysteine of UBE2T and blocking ubiquitin transfer. Biochem.Biophys.Res.Commun., 689:149238-149238, 2023 Cited by PubMed: 37979329DOI: 10.1016/j.bbrc.2023.149238 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.76 Å) |
Structure validation
Download full validation report