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8JIG

A Novel UHRF1-Targeted Compound

Summary for 8JIG
Entry DOI10.2210/pdb8jig/pdb
DescriptorE3 ubiquitin-protein ligase UHRF1, N-[2,4-bis(oxidanylidene)-1H-pyrimidin-5-yl]-N'-oxidanyl-octanediamide (3 entities in total)
Functional Keywordsuhrf1, prostate cancer, dna binding protein
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight48135.70
Authors
Chen, Y.,Jiang, L. (deposition date: 2023-05-26, release date: 2024-05-29)
Primary citationChen, Y.,Jiang, L.
A Novel UHRF1-Targeted Compound
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.4 Å)
Structure validation

222036

PDB entries from 2024-07-03

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