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8J1K

co-crystal structure of non-carboxylic acid inhibitor with PHD2

Summary for 8J1K
Entry DOI10.2210/pdb8j1k/pdb
DescriptorEgl nine homolog 1, N-[(6-cyanopyridin-3-yl)methyl]-5-oxidanyl-2-[(3R)-3-oxidanylpyrrolidin-1-yl]-1,7-naphthyridine-6-carboxamide, MANGANESE (II) ION, ... (4 entities in total)
Functional Keywordsoxidoreductase-inhibitor complex, oxidoreductase/inhibitor
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight24944.22
Authors
Xu, J.,Fu, Y.,Ding, X.,Meng, Q.,Wang, L.,Zhang, M.,Ding, X.,Ren, F.,Zhavoronkov, A. (deposition date: 2023-04-13, release date: 2024-04-17)
Primary citationXu, J.,Fu, Y.,Ding, X.,Meng, Q.,Wang, L.,Man, Z.,Ding, X.,Ren, F.,Zhavoronkov, A.
co-crystal structure of non-carboxylic acid inhibitor with PHD2
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.451 Å)
Structure validation

221051

數據於2024-06-12公開中

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