8IY9
Structure of Niacin-GPR109A-G protein complex
Summary for 8IY9
Entry DOI | 10.2210/pdb8iy9/pdb |
EMDB information | 35817 |
Descriptor | Guanine nucleotide-binding protein G(o) subunit alpha, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... (6 entities in total) |
Functional Keywords | gpcr, g protein, signaling protein |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 5 |
Total formula weight | 147808.49 |
Authors | Yadav, M.K.,Sarma, P.,Chami, M.,Banerjee, R.,Shukla, A.K. (deposition date: 2023-04-04, release date: 2024-03-06, Last modification date: 2024-03-20) |
Primary citation | Yadav, M.K.,Sarma, P.,Maharana, J.,Ganguly, M.,Mishra, S.,Zaidi, N.,Dalal, A.,Singh, V.,Saha, S.,Mahajan, G.,Sharma, S.,Chami, M.,Banerjee, R.,Shukla, A.K. Structure-guided engineering of biased-agonism in the human niacin receptor via single amino acid substitution. Nat Commun, 15:1939-1939, 2024 Cited by PubMed: 38431681DOI: 10.1038/s41467-024-46239-2 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (3.37 Å) |
Structure validation
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