8I0L
Structure of CDK9/cyclin T1 in complex with inhibitor
Summary for 8I0L
Entry DOI | 10.2210/pdb8i0l/pdb |
Descriptor | Cyclin-dependent kinase 9, Cyclin-T1, 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{N},~{N}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide (3 entities in total) |
Functional Keywords | cdk9, inhibitor, complex, cell invasion, cell invasion-inhibitor complex, cell invasion/inhibitor |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 2 |
Total formula weight | 68632.17 |
Authors | |
Primary citation | Jiang, C.,Ye, Y.,Huang, Y. Structure of CDK9/cyclin T1 in complex with inhibitor To Be Published, |
Experimental method | X-RAY DIFFRACTION (3.6 Å) |
Structure validation
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