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8CK5

VDR LBD complex with 25-nitro derivative of 1,25D3

Summary for 8CK5
Entry DOI10.2210/pdb8ck5/pdb
DescriptorVitamin D3 receptor A, Nuclear receptor coactivator 1, ACETATE ION, ... (5 entities in total)
Functional Keywordscomplex, agonist, nuclear receptor, transcription
Biological sourceDanio rerio (zebrafish)
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Total number of polymer chains2
Total formula weight36341.42
Authors
Rochel, N. (deposition date: 2023-02-14, release date: 2023-04-26)
Primary citationGomez-Bouzo, U.,Belorusova, A.Y.,Rivadulla, M.L.,Santalla, H.,Verlinden, L.,Verstuyf, A.,Ferronato, M.J.,Curino, A.C.,Facchinetti, M.M.,Fall, Y.,Gomez, G.,Rochel, N.
Structural analysis and biological activities of C25-amino and C25-nitro vitamin D analogs.
Bioorg.Chem., 136:106528-106528, 2023
Cited by
PubMed: 37054528
DOI: 10.1016/j.bioorg.2023.106528
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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