8BM8

Crystal Structure of Ephrin A2 (EphA2) Receptor Protein Kinase with Compound 11

Summary for 8BM8

• Entry DOI: 10.2210/pdb8bm8/pdb
• Descriptor: Ephrin type-A receptor 2, ~{N}-(3-cyanophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide (3 entities in total)
• Functional Keywords: inhibitor, complex, protein tyrosine kinase, transferase
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 34923.33

Authors

Linhard, V.,Witt, K.,Gande, S.,Wollenhaupt, J.,Lennartz, F.,Weiss, M.S.,Schwalbe, H. (deposition date: 2022-11-10, release date: 2024-06-05)

• Primary citation: Troester, A.; (placeholder, will be filled after publication); To Be Published,

Experimental method

X-RAY DIFFRACTION (1.68 Å)