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8A3A

MTH1 in complex with TH013074

Summary for 8A3A
Entry DOI10.2210/pdb8a3a/pdb
Descriptor7,8-dihydro-8-oxoguanine triphosphatase, 4-(4-methylphenyl)-1~{H}-quinazolin-2-one, SULFATE ION, ... (4 entities in total)
Functional Keywordsnudix, inhibitor, hydrolase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight18586.07
Authors
Liu, H.,Scaletti, E.,Stenmark, P. (deposition date: 2022-06-07, release date: 2023-09-20)
Primary citationLiu, H.,Scaletti, E.,Stenmark, P.
MTH1 in complex with TH013074
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.6 Å)
Structure validation

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