8R5K
The Fk1 domain of FKBP51 in complex with Antascomicine B
Summary for 8R5K
Entry DOI | 10.2210/pdb8r5k/pdb |
Descriptor | Peptidyl-prolyl cis-trans isomerase FKBP5, Antascomicine B (3 entities in total) |
Functional Keywords | isomerase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 14701.93 |
Authors | |
Primary citation | Schafer, S.C.,Voll, A.M.,Bracher, A.,Ley, S.V.,Hausch, F. Antascomicin B stabilizes FKBP51-Akt1 complexes as a molecular glue. Bioorg.Med.Chem.Lett., 104:129728-129728, 2024 Cited by PubMed: 38582133DOI: 10.1016/j.bmcl.2024.129728 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (0.89 Å) |
Structure validation
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