8R4O
Salt inducible kinase 3 in complex with inhibitor
Summary for 8R4O
Entry DOI | 10.2210/pdb8r4o/pdb |
Descriptor | Serine/threonine-protein kinase SIK3, scFvH1, 2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{N}-[(1~{R},2~{S})-2-fluoranylcyclopropyl]-6-methoxy-benzamide, ... (5 entities in total) |
Functional Keywords | kinase inhibitor complex ampk-like salt-induced kinase, ligase |
Biological source | Homo sapiens (human) More |
Total number of polymer chains | 12 |
Total formula weight | 400964.29 |
Authors | |
Primary citation | Oster, L.,Castaldo, M.,de Vries, E.,Edfeldt, F.,Pemberton, N.,Gordon, E.,Cederblad, L.,Kack, H. The structures of salt-inducible kinase 3 in complex with inhibitors reveal determinants for binding and selectivity. J.Biol.Chem., 300:107201-107201, 2024 Cited by PubMed: 38508313DOI: 10.1016/j.jbc.2024.107201 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.725 Å) |
Structure validation
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