8AHG
PAC-FragmentDEL: Photoactivated covalent capture of DNA encoded fragments for hit discovery
Summary for 8AHG
Entry DOI | 10.2210/pdb8ahg/pdb |
Descriptor | Serine/threonine-protein kinase PAK 4, ~{N}-methyl-3-propan-2-yl-1~{H}-pyrazolo[3,4-c]pyridine-4-carboxamide (3 entities in total) |
Functional Keywords | protein kinase, pak4, atp-binding, transferase, technology |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 33599.00 |
Authors | Baker, L.M.,Murray, J.B.,Hubbard, R.E. (deposition date: 2022-07-21, release date: 2022-09-14, Last modification date: 2024-01-31) |
Primary citation | Ma, H.,Murray, J.B.,Luo, H.,Cheng, X.,Chen, Q.,Song, C.,Duan, C.,Tan, P.,Zhang, L.,Liu, J.,Morgan, B.A.,Li, J.,Wan, J.,Baker, L.M.,Finnie, W.,Guetzoyan, L.,Harris, R.,Hendrickson, N.,Matassova, N.,Simmonite, H.,Smith, J.,Hubbard, R.E.,Liu, G. PAC-FragmentDEL - photoactivated covalent capture of DNA-encoded fragments for hit discovery. Rsc Med Chem, 13:1341-1349, 2022 Cited by PubMed: 36426238DOI: 10.1039/d2md00197g PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.885 Å) |
Structure validation
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