7VTO

The crystal structure of PAK1 with the inhibitor GW8510

Summary for 7VTO

• Entry DOI: 10.2210/pdb7vto/pdb
• Descriptor: Serine/threonine-protein kinase PAK 1, 4-[(7-OXO-7H-THIAZOLO[5,4-E]INDOL-8-YLMETHYL)-AMINO]-N-PYRIDIN-2-YL-BENZENESULFONAMIDE (3 entities in total)
• Functional Keywords: pak1, inhibitor, complex, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 2
• Total formula weight: 68206.07

Authors

Zhu, S.J. (deposition date: 2021-10-30, release date: 2022-11-02, Last modification date: 2023-11-29)

• Primary citation: Zhu, S.J.; The crystal structure of PAK1 with the inhibitor GW8510; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.59 Å)