7T39
Co-crystal structure of human PRMT9 in complex with MT221 inhibitor
7T39 の概要
エントリーDOI | 10.2210/pdb7t39/pdb |
分子名称 | Protein arginine N-methyltransferase 9, 7-[5-S-(4-{[(2-ethylpyridin-3-yl)methyl]amino}butyl)-5-thio-beta-D-ribofuranosyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine (3 entities in total) |
機能のキーワード | methyltransferase, prmt9, sgc, structural genomics, structural genomics consortium, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
由来する生物種 | Homo sapiens (human) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 80958.90 |
構造登録者 | Zeng, H.,Dong, A.,Hutchinson, A.,Seitova, A.,Li, Y.,Gao, Y.D.,Schneider, S.,Siliphaivanh, P.,Sloman, D.,Nicholson, B.,Fischer, C.,Hicks, J.,Brown, P.J.,Arrowsmith, C.H.,Edwards, A.M.,Halabelian, L.,Structural Genomics Consortium (SGC) (登録日: 2021-12-07, 公開日: 2021-12-22, 最終更新日: 2023-10-18) |
主引用文献 | Zeng, H.,Dong, A.,Hutchinson, A.,Seitova, A.,Li, Y.,Gao, Y.D.,Schneider, S.,Siliphaivanh, P.,Sloman, D.,Nicholson, B.,Fischer, C.,Hicks, J.,Brown, P.J.,Arrowsmith, C.H.,Edwards, A.M.,Halabelian, L.,Structural Genomics Consortium (SGC) Co-crystal structure of human PRMT9 in complex with MT221 inhibitor To Be Published, |
実験手法 | X-RAY DIFFRACTION (2.81 Å) |
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