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7SMP

CryoEM structure of NKCC1 Bu-I

Summary for 7SMP
Entry DOI10.2210/pdb7smp/pdb
EMDB information25204
DescriptorSolute carrier family 12 member 2, 3-(butylamino)-4-phenoxy-5-sulfamoylbenzoic acid, POTASSIUM ION (3 entities in total)
Functional Keywordscotransporter, dimer, ion, membrane protein, transport protein
Biological sourceHomo sapiens (human)
Total number of polymer chains2
Total formula weight207798.29
Authors
Moseng, M.A. (deposition date: 2021-10-26, release date: 2022-09-28, Last modification date: 2023-05-31)
Primary citationMoseng, M.A.,Su, C.C.,Rios, K.,Cui, M.,Lyu, M.,Glaza, P.,Klenotic, P.A.,Delpire, E.,Yu, E.W.
Inhibition mechanism of NKCC1 involves the carboxyl terminus and long-range conformational coupling.
Sci Adv, 8:eabq0952-eabq0952, 2022
Cited by
PubMed: 36306358
DOI: 10.1126/sciadv.abq0952
PDB entries with the same primary citation
Experimental method
ELECTRON MICROSCOPY (3.28 Å)
Structure validation

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