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7REL

Crystal structure of the first bromodomain (BD1) of human BRD4 in complex with dual BRD4-JAK2 inhibitor MA9-060

Summary for 7REL
Entry DOI10.2210/pdb7rel/pdb
DescriptorBromodomain-containing protein 4, 1,2-ETHANEDIOL, N-[2-chloro-5-({2-[3-fluoro-4-(1-methylpiperidin-4-yl)anilino]-5-methylpyrimidin-4-yl}amino)phenyl]-2-methylpropane-2-sulfonamide, ... (4 entities in total)
Functional Keywordsbet, jak2, dual brd-kinase inhibitor, gene regulation
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight15722.56
Authors
Karim, M.R.,Schonbrunn, E. (deposition date: 2021-07-13, release date: 2021-07-21, Last modification date: 2023-10-18)
Primary citationKarim, M.R.,Schonbrunn, E.
Crystal structure of the first bromodomain (BD1) of human BRD4 in complex with dual BRD4-JAK2 inhibitor MA9-060
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.55 Å)
Structure validation

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