7QGE
H. SAPIENS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 5,6,7,8-TETRABROMOBENZOTRIAZOLE (TBBt) AT PH 8.5
Summary for 7QGE
Entry DOI | 10.2210/pdb7qge/pdb |
Related | 6TLL 6TLP |
Descriptor | Casein kinase II subunit alpha, 4,5,6,7-TETRABROMOBENZOTRIAZOLE, CHLORIDE ION, ... (5 entities in total) |
Functional Keywords | ck2, casein kinase 2, inhibitor, bromo-benzotriazole, halogen bond, transferase-inhibitor complex, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 46855.98 |
Authors | Winiewska-Szajewska, M.,Czapinska, H.,Kaus-Drobek, M.,Piasecka, A.,Mieczkowska, K.,Dadlez, M.,Bochtler, M.,Poznanski, J. (deposition date: 2021-12-08, release date: 2022-10-19, Last modification date: 2024-01-31) |
Primary citation | Winiewska-Szajewska, M.,Czapinska, H.,Kaus-Drobek, M.,Fricke, A.,Mieczkowska, K.,Dadlez, M.,Bochtler, M.,Poznanski, J. Competition between electrostatic interactions and halogen bonding in the protein-ligand system: structural and thermodynamic studies of 5,6-dibromobenzotriazole-hCK2 alpha complexes. Sci Rep, 12:18964-18964, 2022 Cited by PubMed: 36347916DOI: 10.1038/s41598-022-23611-0 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.27 Å) |
Structure validation
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