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7PQS

SRPK1 in complex with MSC2711186

Summary for 7PQS
Entry DOI10.2210/pdb7pqs/pdb
DescriptorSRSF protein kinase 1, ~{N}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{H}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{N}-methyl-methanesulfonamide, GLYCEROL, ... (8 entities in total)
Functional Keywordskinase, inhibitor, complex, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight88748.40
Authors
Schroeder, M.,Leiendecker, M.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2021-09-20, release date: 2021-12-15, Last modification date: 2024-01-31)
Primary citationSchroeder, M.,Leiendecker, M.,Knapp, S.
SRPK1 in complex with MSC2711186
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

250835

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