7LL5
High-resolution crystal structure of human JAK2 kinase domain (JH1) bound to PN5-150.
Summary for 7LL5
Entry DOI | 10.2210/pdb7ll5/pdb |
Descriptor | Tyrosine-protein kinase JAK2, 1,2-ETHANEDIOL, {1-(ethylsulfonyl)-3-[4-(2-{[4-(1-methylpiperidin-4-yl)phenyl]amino}-7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]azetidin-3-yl}acetonitrile, ... (4 entities in total) |
Functional Keywords | rheumatoid arthritis, innate immuninity, adaptive immunity, myeloproliferative neoplasms, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 35120.13 |
Authors | Karim, M.R.,Schonbrunn, E. (deposition date: 2021-02-03, release date: 2022-01-12, Last modification date: 2023-11-15) |
Primary citation | Karim, M.R.,Schonbrunn, E. High-resolution crystal structure of human JAK2 kinase domain (JH1) bound to PN5-150. To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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